AG-120 (racemic) ( —— )

产品货号. M23614 CAS No. 1448346-63-1

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

AG-120 (racemic)
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

AG-120 (racemic), the racemic mixture of AG-120, is an orally available isocitrate dehydrogenase type 1 (IDH1) inhibitor, and shows potential antineoplastic activity.
产品描述

AG-120 (racemic), the racemic mixture of AG-120, is an orally available isocitrate dehydrogenase type 1 (IDH1) inhibitor, and shows potential antineoplastic activity.
同义词

——
通路

Metabolic Enzyme/Protease
靶点

Dehydrogenase
受体

IDH1
研究领域

——
适应症

——

CAS Number

1448346-63-1
分子量

583.0
分子式

C28H22ClF3N6O3
纯度

>98% (HPLC)
溶解度

DMSO:100 mg/ml (171.54 mM); Ethanol:100 mg/ml (171.54 mM)
SMILES

O=C1CC[C@@H](C(N(C(C(NC2CC(F)(F)C2)=O)C3=CC=CC=C3Cl)C4=CC(F)=CN=C4)=O)N1C5=NC=CC(C#N)=C5
化学全称

——

1.M Cecilia Caino, Dario C Altieri. Clin Cancer Res. 2016 Feb 1;22(3):540-5.

计算器

产品手册

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